Affordable Access

Publisher Website

A new and efficient procedure for preparing 1,2,3-triazoles

Authors
Journal
Tetrahedron Letters
0040-4039
Publisher
Elsevier
Publication Date
Volume
38
Issue
29
Identifiers
DOI: 10.1016/s0040-4039(97)01137-4

Abstract

Abstract 1,2,3-Triazoles are readily accessible in moderate to good yields by a diazo transfer reaction with β-amino-α,β-unsaturated ketones or esters and tosyl or mesyl azide reagent. In this methodology the nitrogen atoms N-2 and N-3 of the triazole ring are derived from diazo transfer reagent and nitrogen atom N-1 is derived from the appropriate enamine.

There are no comments yet on this publication. Be the first to share your thoughts.