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Concise synthesis of aromatic tertiary amines via a double Petasis–borono Mannich reaction of aromatic amines, formaldehyde, and organoboronic acids

Authors
Journal
Tetrahedron Letters
0040-4039
Publisher
Elsevier
Volume
55
Issue
29
Identifiers
DOI: 10.1016/j.tetlet.2014.03.131
Keywords
  • Petasis–Borono Mannich Reaction
  • Organoboronic Acids
  • Aromatic Amines
  • Formaldehyde
  • Multi-Component Reaction

Abstract

Graphical abstract A simple and efficient strategy to construct aromatic tertiary amines via a double Petasis–borono Mannich reaction of aromatic amines, formaldehyde and organoboronic acids has been developed. The transformation provides a useful method for the synthesis of amine derivatives.

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