Li, Zhenxing Yang, Binxin Ding, Yue Meng, Jiao Hu, Jinhong Zhou, Xiang Liu, Liwei Wu, Zhibing Yang, Song
Published in
International journal of biological macromolecules
Plant diseases caused by malignant and refractory phytopathogenic viruses have considerably restricted crop yields and quality. To date, drug design targeting functional proteins or enzymes of viruses is an efficient and viable strategy to guide the development of new pesticides. Herein, a series of novel eugenol derivatives targeting the tobacco m...
Van Thong, Pham; Van Meervelt, Luc; 14577; Chi, Nguyen Thi Thanh;
status: published
Muniz, Débora Feitosa Dos Santos Barbosa, Cristina Rodrigues de Menezes, Irwin Rose Alencar de Sousa, Erlânio Oliveira Pereira, Raimundo Luiz Silva Júnior, João Tavares Calixto Pereira, Pedro Silvino de Matos, Yedda M L S da Costa, Roger H S de Morais Oliveira-Tintino, Cícera Datia...
...
Published in
Food chemistry
Staphylococcus aureus is a Gram-positive bacterium responsible for a number of diseases and has demonstrated resistance to conventional antibiotics. This study aimed to evaluate the antibacterial activity of eugenol and its derivatives allylbenzene, 4-allylanisole, isoeugenol and 4-allyl-2,6-dimethoxyphenol against the S. aureus NorA efflux pump (E...
Dhiman, Priyanka Malik, Neelam Khatkar, Anurag
Published in
BMC Chemistry
Natural based inhibitors of monoamine oxidase are promising drug candidates for the treatment of several neurodegenerative and neuropsychological disorders including depression, anxiety, Parkinson’s disease and Alzheimer’s disease. In the present study we designed and synthesized the eugenol based derivatives and investigated them for human MAO inh...
Vargas-Méndez, Leonor Y Sanabria-Flórez, Pedro L Saavedra-Reyes, Laura M Merchan-Arenas, Diego R Kouznetsov, Vladimir V
Published in
Saudi journal of biological sciences
The anti-acetylcholinesterase, larvicidal, antifeedant activities and general toxicity of 15 semisynthetic eugenol derivatives based on clove oil (including the own oil), were evaluated against the maize armyworm, Spodoptera frugiperda (J.E. Smith). Therefore, promising eugenol molecules were classified with larvicidal, anti-acetylcholinesterase an...
de Souza, Thiago Belarmino Orlandi, Marina Coelho, Luiz Felipe Leomil Malaquias, Luiz Cosme Cotta Dias, Amanda Latercia Tranches de Carvalho, Roberta Ribeiro Silva, Naiara Chaves Carvalho, Diogo Teixeira
Published in
Medicinal Chemistry Research
Six eugenol glycosides were prepared in order to assess their antifungal activity against Candida species. They were synthesized by glycosylation of eugenol with the appropriate glycosyl bromides followed by deacetylation with sodium methoxide in methanol and were evaluated in vitro for their antifungal activity through a Mueller–Hinton broth micro...
Wang, Xinlong Yi, Meigui Du, Quanhai Wu, Aimin Xiao, Rong
Published in
Medicinal Chemistry Research
A novel series of pyrethriods was designed and synthesized by connecting various eugenol derivatives to either a chrysanthematic acid or 2-(4-chlorophenyl)-3-methylbutanoic acid. The insecticidal activity of target compounds has been evaluated by an immersion method on the fourth instar larvae of Culex pipens quinquefasciatus. The results revealed ...
